Thanzi, Kukonzekera
"Dorzopt" (m'maso): zimatsogolera ndemanga, analogs
Khungu - gulu m'malo lalikulu la matenda diso, amene yodziwika ndi nthawi kapena okhazikika kuwonjezeka kuthamanga intraocular ndi zilema wotsatira chitukuko, chamawonedwe manja ndi kuchepa acuity zithunzi.
Zochizira matenda pogwiritsa ntchito mankhwala osiyana. The mankhwala ambiri ndi "Dorzopt" (diso madontho). Ogula ndemanga, malangizo pa ntchito mankhwala amenewa ayankhidwa pansipa.
Kulongedza katundu ndi zikuchokera
Kodi mankhwala lili mankhwala "Dorzopt" (diso madontho)? The yogwira zikuluzikulu za mankhwala ndi dorzolamide (monga hydrochloride). Ndiponso medicament lili zotsatirazi zinthu wothandiza: Benzalkonium enaake, gietelloza, mannitol, hydroxide sodium, citric acid monohydrate, madzi oyera.
Ankaona mankhwala opangidwa mu mbale polyethylene ndi 5 ml dropper nozzle.
pharmacodynamics
Kodi m'maso "Dorzopt"? Guide inanena kuti chida ichi ndi m'dera carbonic anhydrase woletsa. Iwo ali kumafooketsa pa intraocular katulutsidwe madzimadzi ndi kumabwezera mmbuyo mapangidwe carbonate hydrogen ndi madzi imafoola kulanda ndi sodium wochuluka.
Izi mankhwala sayambitsa miosis kapena khungu usiku, komanso kuphipha wa malawi.
Pharmacokinetics
ngati mankhwala imatsala, "Dorzopt" (diso madontho)? Mayamwidwe mankhwala kumachitika mwa diso ndi kupyolera mu nthambi ndi sclera. mankhwala zokhudza zonse mitengo mayamwidwe ndi otsika.
Kamodzi m'magazi, mankhwala yogwira pophika mofulumira likulowerera ku maselo ofiira ndi okhutira mkulu wa carbonic anhydrase 2.
Kulankhulana ndi mapuloteni plasma amapezeka ndi 33%. mankhwala ndi kutembenukira ku N-dezetilirovanny metabolite, amene si wokangalika ndi carbonic anhydrase 2, koma amatha kutsekereza wina carbonic anhydrase.
ntchito yaitali mankhwala kumabweretsa kudzikundikira zake erythrocytes.
Anasonyeza mankhwala kudzera impso. kuchotsa awo ali 2 Kupha gawo: kudya ndi pang'onopang'ono. inawo chifukwa cha pang'onopang'ono kutuluka kwa yogwira chigawo maselo a magazi.
theka moyo nthawi za 4 months.
umboni
Pamene prescribers "Dorzopt"? Diso madontho zimathandiza kwambiri pa matenda a okwera intraocular kuthamanga pa anthu ndi oopsa ocular kapena otsegula pseudoexfoliative khungu (kuphatikizapo sekondale).
contraindications
Kodi milandu, simungathe ntchito mankhwala "Dorzopt"? madontho diso si analamula kuti:
- hyperchloraemic acidosis;
- Hypersensitivity nyengo constituent;
- matenda a impso chaukali;
- ngati mwana;
- mu nthawi ya mkaka wa m'mawere.
Ndi kusamala kwambiri ayenera kugwiritsidwa ntchito chida ichi:
- shuga;
- odwala ndi kuwonongeka kwa chiwindi;
- anthu kachulukidwe ka maselo diso endothelium diso (a Mwina mkulu wa edema corneal).
dosing
Perekani chida wosasamala zochizira matenda diso ali yekha katswiri yopapatiza ndikatha kumfunsafunsa kusamala wodwala. Kwirirani chiphunzitso desirably dontho limodzi mu za sac conjunctival wa katatu patsiku.
Ndi osakaniza mankhwala ndi beta-blockers apakhungu mankhwala ntchito dontho limodzi kawiri pa tsiku.
Ngati ocular matenda mankhwala zikuphatikizapo wothandizila angapo ophthalmic, ndi imeneyi pakati instillation awo ayenera kukhala mphindi zosachepera khumi.
zotsatira zoyipazi
Ngati inu ntchito m'maso "Dorzopt" otsatirawa zosiyanasiyana m'dera angathe odwala:
- Kuyabwa ndi moto kumverera mu maso, conjunctivitis, paresthesia, chikope edema, pom'ng'amba, blepharitis, mkhutu momveka za masomphenya, photophobia ndi kungotengeka punctate keratitis.
- kawirikawiri ndi kugwiritsa ntchito mankhwala ndi: iridocyclitis, kuwonjezera makulidwe a diso, ziwengo, hypotension diso ndi retinal detachment pambuyo ntchito antiglaukomatoznyh.
zotsatira zokhudza zonse mbali:
- kumverera kwa nseru, kulawa zowawa m'kamwa, chitukuko nefrourolitiaza, kutopa, migraine, zilonda exudative erythema multiforme, poizoni epidermal necrolysis, aplastic magazi, zotupa pa khungu ndi agranulocytosis.
Nthawi cha mankhwala osokoneza bongo
Kodi zizindikiro zikayamba ntchito "Dorzopt" mlingo waukulu wa mankhwala? Eyedrops, analogs amene ali pansipa, angathandize:
- acidosis chitukuko;
- kusokonezeka kwa madzi ndi bwino electrolyte;
- CNS mavuto.
Zochizira wotere ntchito symptomatically, limodzi ndi ulamuliro wa mlingo wa electrolytes ndi magazi pH.
Mwanjira mankhwala
- Pamene pamodzi ndi wothandizila mankhwala antiglaucoma (beta-blockers, "dipivefrin", "pilocarpine", "Carbachol") amakulitsa zotsatira zake.
- Ndi "acetazolamide" kumaonjezera ngozi ya zotsatira zokhudza zonse mbali.
- Ndi Mlingo zikuluzikulu asidi acetylsalicylic kumawonjezera kawopsedwe wa mankhwala.
ayamikira yeniyeni
The ntchito mbale multidose mwina hule chitukuko cha keratitis bakiteriya. Ichi ndi chifukwa kuipitsidwa inadvertent za nthanoyi.
Pa mankhwala "Dorzoptom" sayenera kugwiritsa ntchito magalasi monga benzalkonium mankhwala enaake angakhale oopsa ndi kuyambitsa kuyabwa ndi maso.
Analogs ndi mtengo mankhwala
Sinthanitsani mankhwala ankaona kuti diso silingathe kudzera monga "Trusopt" ndi "Floksal". Mtengo wa mankhwala ndi za 350 rubles.
ndemanga ogula
Mwatsoka, ogula ndemanga za mankhwala "Dorzopt" n'zochepa. Mwa ubwino waukulu chidwi imeneyi mankhwala monga kupezeka ndi moyenerera. Komabe, ena ogula nkhawa, m'dera ndi zokhudza zonse zosiyanasiyana chokhwima komwe kumachitika nthawi chithandizo ndi madontho. Pankhani imeneyi, akatswiri akhoza kulengeza ntchito mankhwala pansi pa dzina "Dorzopt Plus".
Eyedrops tatchulazi Zina mankhwala zina, monga timolol. Iwo amalimbitsa ngalande za madzimadzi intraocular.
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