ThanziKukonzekera

Miyala 'Eufillin': zikuonetsa ntchito

"Eufillin" Mapale ndi Adenozinergicheskie njira, ndi ofanana ndi "aminophylline Escom," "Aminofilliin" "Euffillin-Darnitsya". Waukulu yogwira mankhwala yokonza pamwamba akutumikira aminophylline ndi wocheperapo - asidi stearic ndi wowuma mbatata.

"Eufillin": ikulongosola za mankhwala

Izi mankhwala ali zimakhudzanso ntchito zosiyanasiyana za thupi. Eufillin kumapangitsa chapakati mantha dongosolo, kumaonjezera contractile myocardium ntchito, amachititsa patsogolo aimpso, inatsekeratu ndi zotumphukira mitsempha, kumathandiza kuthamanga mu mtsempha wamagazi ndi m'mapapo mwanga kuchepetsa, ndipo kwambiri kumawonjezera aimpso magazi. Komanso, "Eufillin" miyala ndi zolimbitsa diuretic zotsatira, ziletsa kupatsidwa zinthu za m'mwazi loitanirana, ziletsa amasulidwe mlongoti selo instigators ziwengo. Iwo amachepetsa contractile ntchito minofu yosalala, chotero Masulani bronchial machubu ndi kuchotsa bronchospasm. Anati kukonzekera bwino chosakanikirana ndi ndende wake pazipita mu magazi kumachitika mwa maora awiri makonzedwe, koma Komabe, nawonso kudya metabolised ndi chiwindi, kumene metabolites anafooka anapanga. About 10% ya mankhwala analandira excreted zikutsatiridwa mu mkodzo.

Miyala "Eufillin": a zikuonetsa

mankhwala cholinga ntchito pamaso pa bronchospasm ndi mphumu, mphumu mtima, matenda oopsa kunachitika kufalitsa m'mapapo mwanga, ngati kuukira limodzi bronchospasm ndi matenda kupuma wa Cheyne-Stokes. Iwo ntchito mu nkhani ya kufunika aziyenda bwino oziziritsa ndi mpumulo wa mavuto oziziritsa mtima, iwo kuchepetsa kuthamanga intracranial, edema oziziritsa, zimachitika mu sitiroko ischemic kapena pamene walephera aakulu a kapezedwe magazi ku ubongo.

"Eufillin" mapiritsi: malangizo ntchito mankhwala

Mankhwala akutengedwa pakamwa, pambuyo chakudya, nthawi imodzi katatu pa tsiku mlingo wa akuluakulu ndi magalamu 0,15. Mlingo umodzi kwa mtima wamkulu mwina upambana 0,5 ga Ana analandira kukonzekera mlingo yafupika 7-10mg / kg ndi alipire Mlingo 4 pa tsiku. Ana mu sitepe imodzi mlingo umodzi sangakhale kuposa 7 mg / kg.

Ngati kusowa kwa ntchito za machitidwe biotransformation enzyme a chiwindi odwala pa zaka 55 ndi neonates, mankhwala "Eufillin" anatumizidwa mosamala kwambiri.

Mankhwalawo amene amayambitsa miyala "Eufillin"

Mukalola phwando wothandizila pa chopanda kanthu m'mimba, zingaoneke zizindikiro dyspeptic, amene kugwirizana ndi mtima mankhwala katundu. Komanso pa nkhani ya tilinazo mkulu ethylenediamine kumachitika dermis exfoliative kapena febrile anachita.

contraindications

Kugwiritsa ntchito mankhwala ndi contraindicated mu khunyu, hypotension kwambiri, arrhythmia ndi tachycardia paroxysmal. Musawachite mapiritsi "Eufillin" pamaso pa kulephera mtima, makamaka ngati amagwirizana ndi infarction m'mnyewa wamtima, komanso pamene pali mtima mungoli matenda, kapena inatsekeratu insufficiency.

Ambiri osokoneza "Eufillin"

Mu chochitika cha mankhwala osokoneza bongo pali zizindikiro monga kutsekula m'mimba, kupweteka epigastric, anorexia, magazi m'mimba, kunyansidwa, m'chikaiko chowakaikitsa, tachycardia, zowombetsa mkota khunyu, arrhythmia yamitsempha yamagazi, ankatenthetsa nkhope, kusanza, kugona, hipnoe ndi photophobia.

Mu milandu, muyenera yomweyo isiye kugwiritsa ntchito mankhwala "Eufillin" ndi kuyamba yotithandiza excretion wake ku thupi, amene n'kofunika kusamba kunja m'mimba gwirani amakakamizidwa diuresis, hemosorption, plasmasorption, hemodialysis, peritoneal dialysis, ndi chithandizo ndiye symptomatic.

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