Thanzi, Kukonzekera
Kugwiritsa antispasmodic "Papaverine Hydrochloride"
Kukonzekera "Papaverine hydrochloride" amatanthauza miotropnym njira kolimbikira spasmolytic kwenikweni. Kwa zaka zambiri, amagwiritsidwa ntchito kuchepetsa mtima kamvekedwe ndi minofu yosalala zosangalatsa ndipo pafupifupi onse ziwalo. Iwo ali kutchulidwa kanthu hypotensive. Izi mankhwala dilates mitsempha, kumawonjezera magazi buku, makamaka ubongo. Izi mankhwala mu mlingo waukulu kwambiri amachepetsa excitability minofu mtima, komanso kumathandiza kuti liwiro intracardiac madutsidwe. mphamvu zake pa chapakati mantha dongosolo chimaoneka pang'ono, ngakhale kuti ali ndi zotsatira sedative pa mlingo waukulu.
Kumasulidwa kukonzekera "Papaverine hydrochloride" m'njira ngati mlingo:
- mapiritsi akuluakulu 0,04g (10 ma PC.);
- mapiritsi Ana a 0.01g (10 ma PC.);
- 2% jekeseni (10 ampoules);
- thumbo suppositories 20 mg (10 ma PC.).
Zikuonetsa ntchito ndi zinthu monga kuphipha ziwalo yosalala minofu peritoneum cholecystitis, aimpso colic; chonsechi matenda a m'matumbo; endarteriite; bronchospasm; pilorospazme; mtima spasms, ili mu ubongo. Mankhwalawa angina pectoris amatanthauza "Papaverine Hydrochloride" ntchito ophatikizana mankhwala ndi mankhwala ena.
Contraindications ntchito mankhwala awa:
hypersensitivity, mkhutu chiwindi ntchito, khungu, ubwana (zaka 0.5). Okalamba sayenera kumwa mankhwala chifukwa cha chiopsezo hyperthermia.
Amatanthauza "Papaverine hydrochloride": malangizo ntchito
mankhwala ikuchitika kwa 3-4 p. patsiku. Mlingo wa utsogoleli umodzi miyala zimasiyanasiyana ndi zaka wodwalayo. Akuluakulu anaika miyala mlingo umodzi 40-60mg. Ana 0.5-2 ga - 5mg, 3-4 PM - 5-10mg, 5-6 L. -10mg, 7-9 malita. - 10-15mg, 10-14 malita. - 15-20mg.
Jekeseni chikuyendetsedwera intramuscularly kapena subcutaneously. Majekeseni kuchita 2-4 p. pa tsiku ndi 1-2ml. Mtsempha mankhwala jekeseni pang'onopang'ono pa 20mg kale kuwonjezera thereto sodium kolorayidi 10-20ml (0.9% njira). Ndondomeko bwino ikuchitika kuyang'aniridwa ndi dokotala. Kwa odwala zaka umodzi mlingo woyambilira sayenera upambana 10 mg. Nthawi zambiri mankhwala chikuyendetsedwera parenterally limodzi ndi mankhwala osiyanasiyana spazmaliticheskimi ndi analgesic, monga mankhwala "Promedol".
Makandulo ndi papaverine kutumikiridwa rectally, 2-3 p. 20-40mg pa tsiku.
Kukonzekera "Papaverine hydrochloride" Mwina kuyambitsa zotsatira zoyipa monga kugona, thupi lawo siligwirizana, arrythmia yamitsempha yamagazi, upregulation wa transaminases chiwindi, kutsitsa magazi, kudzimbidwa, eosinophilia.
Ngati zizindikiro ambiri osokoneza anati monga kufooka ambiri, diplopia, hypersomnia.
Mwa kugwiritsa ntchito malangizo wapadera umenewu kuchita mankhwala amalangiza ntchito mosamala mankhwala chakhungu odwala ndi okalamba; anthu ndi kuvulala mutu, hypothyroidism, dysfunctions adrenal, impso ndi chiwindi; tachycardia; zinthu mantha.
Mankhwala "Papaverine hydrochloride" pa mimba ndi pamene akudya ndi bwino ntchito chifukwa cha kugwira kwake ndi chitetezo nthaŵi si anaika.
Pa mankhwala mowa ndikoletsedwa. Kusuta pa chithandizo kwambiri amachepetsa mphamvu ya mankhwala. Pamodzi ndi kuvomereza amatanthauza "Papaverine" ndi "Dopegitom" Chinthu choyamba ndi kwambiri yafupika.
Papaverine hydrochloride ali m'gulu angapo ophatikizana MANKHWALA OLETSA VUTOLI osakaniza ndi zinthu zina mankhwala:
- mankhwala "Lyupaverin" - ndi phenobarbital;
- mankhwala "Pafillin" - ndi platifillin gidrotata;
- kukonzekera "Kellatrin" - ndi kellinu ndi atropine sulphate ;
- mankhwala "Kelliverin" - ndi Kellin;
- kukonzekera "Nikoverin" - acid nicotinic.
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