Thanzi, Kukonzekera
"Tsinarin": malangizo ntchito kwenikweni Anzawo
blockers kashiamu njira otchedwa sakanikira gulu la mankhwala ndi chimodzimodzi opaleshoni mfundo, koma amasiyana ena katundu, kuphatikizapo magawo kayendedwe, minofu selectivity ndi zotsatira pa mlingo mtima.
Mfundo zikuluzikulu za ntchito mankhwala amenewa ndi amene amatha ziletsa malowedwe a Ca ayoni kwa danga extracellular m'zotengera magazi ndi maselo mtima minofu kudzera njira kashiamu (m'mbuyo). Zimenezi zimabweretsa kutchulidwa vasodilator kanthu.
Wotchuka kwambiri kashiamu antagonist ndi mankhwala "tsinarin". Malangizo ntchito, mtengo, ndi ndemanga zikuchokera ndalama adzakhala pansipa.
kumasulidwa mawonekedwe, ma CD, maonekedwe, zikuchokera
Mankhwala "tsinarin", ndemanga zimene ziri zabwino, iwo akugulitsa mawonekedwe a biconvex, kuzungulira ndi miyala woyera. chigawo chawo chachikulu ndicho cinnarizine. Kupatula izo, zikuchokera mankhwala limapangidwa monga excipients povidone K25, lactose, wowuma tirigu, colloidal pakachitsulo woipa ndi magnesium stearate.
Izi zikutanthauza mugule maselo a mizere.
makhalidwe mankhwala
pa ntchito "tsinarin" mankhwala Guide ikusimba kuti antagonist kusankha njira kashiamu (m'mbuyo). Amachepetsa otaya Ca ion ku maselo amachepetsa chiwerengero plasmolemma zofikira, komanso timapitiriza vasodilating zotsatira za mpweya woipa komanso amachepetsa minofu kamvekedwe ka arterioles lapansi.
Tikamachita zinthu mwachindunji pa zotengera, mankhwala kwambiri kumachepetsa kubvomereza kwawo kwa zakudya (norepinephrine, Epinephrine, angiotensin, vasopressin, ndi dopamine). Komanso dziwani kuti medicament ankaona ali vasodilating katundu, kuphatikizapo ndi ziwiya ubongo. Pankhaniyi, izo ziribe mphamvu pa magazi.
Mankhwala "tsinarin", mtengo wa amene alembedwa pansipa, ndi amtengo kutchulidwa ntchito mankhwala a antihistamine, izo kumachepetsa excitability wa zida za vestibular ndipo kumachepetsa kamvekedwe wa NS chisoni. Izi mankhwala bwino khalidwe ngati koyamba cerebrovascular insufficiency ndi aakulu. Anthu ndi mkhutu kufalitsidwa zotumphukira bwino magazi kuti zimakhala onse ndi ziwalo. Ndi njira kuchepetsa kukhuthala magazi, kumaonjezera elasticity wa Kakhungu maselo a magazi ndi minofu kukana kuti hypoxia.
The kinetics wa mankhwala
mbali Kodi kayendedwe chibadidwe mankhwala "tsinarin"? Malangizo Ntchito limanena kuti wothandizila izi resorbed mu matumbo ndi m'mimba. Pachimake plasma ndende akwaniritsa pambuyo maola atatu. Kulankhulana ndi cinnarizine plasma mapuloteni ndi 91%. mankhwala kwathunthu zimapukusidwa mu chiwindi. theka moyo wake nthawi maola anayi. Likukhalira mankhwala mu mkodzo ndi ndowe.
umboni
Mankhwala "tsinarin" akusonyeza phwando:
- senile maganizo;
- ischemic sitiroko;
- cranial mabvuto;
- zinthu pambuyo sitiroko (kuphatikizapo mu hemorrhagic sitiroko);
- mtima encephalopathy;
- kwa kinetoses prophylaxis (apanyanja kapena matenda mpweya, komanso pa akugwedeza);
- matenda vestibular (kuphatikizapo ndi matenda Meniere a, tinnitus, vertigo, nystagmus, kusanza ndi nseru chiyambi labyrinthine);
- migraine (popewa kuukira);
- kuphwanya makope zotumphukira.
Contraindications kulandira magomewo
Kodi zinthu sayenera mankhwala mankhwala "tsinarin"? Malangizo malipoti ntchito kuti mankhwala awa contraindicated mu:
- hypersensitivity;
- gestation;
- yoyamwitsa.
Iwo ayenera kukumbukira kuti mankhwala Kwalamulidwa mosamala matenda Parkinson.
Mankhwala "tsinarin": malangizo ntchito
Pakumwa mapiritsi tiziiona mkati, makamaka pambuyo chakudya.
Pamene maganizo, kufalitsa mankhwala ubongo magazi kutumikiridwa mu kuchuluka kwa 25-50 mg wa katatu pa tsiku, ndi zotumphukira magazi - pa 50-75 mg wa ndi multiplicity chomwecho.
Pamene matenda vestibular analimbikitsa kutenga mankhwala pa 25 mg katatu patsiku. Pamene kinetosis kapena otchedwa "njira" wamkulu odwala matenda kutumikiridwa 25 mg wa mankhwala kwa mphindi 30 asanayambe ulendo. Ngati chofunika, mankhwala atapatsidwa mobwerezabwereza pambuyo maola 6 (mu yofanana).
Ana, mankhwala Kwalamulidwa kuchuluka kwa 1/2 mlingo wamkulu.
Pa mkulu kudziwa mankhwala medicament akuyamba ndi theka mlingo pang'onopang'ono kuonjezera. The njira ya mankhwala ukhoza kulikonse kwa masabata 2-3 miyezi ingapo.
zotsatira zoyipazi
Izi mankhwala zikhoza zotsatirazi zochita mbali:
- youma pakamwa, dyspepsia, epigastric ululu, cholestatic matenda a chikasu ndiyo;
- kusinza, litsipa, kutopa, ndi matenda extrapyramidal (mwachitsanzo, kuchuluka minofu kamvekedwe, kugwedeza wa miyendo hypokinesia);
- ndere planus, thukuta, lupus-monga matenda, zotupa pa khungu;
- Zotsatira siligwirizana, kunenepa kwambiri, utachepa magazi.
Price, tchuti analogues mankhwala ndi ndemanga za izo
Yopereka mankhwala cha gulu limeneli la blockers kashiamu njira, kuyendetsedwa ndi mankhwala dokotala. Mtengo wa mankhwala ndi za 20-50 rubles.
Ngati ndi kotheka, chida akhoza m'malo mankhwala "Vertizin", "Diziron", "Stugezin", "stugeron", "Tsinazin", "Tsinedil" "Cinnarizine" ndi zina zotero.
ogula ambiri akutenga antagonist uyu amati ndi kothandiza kwambiri komanso zothandiza mankhwala. Mankhwala "tsinarin" amathandiza kuthetsa matenda vestibular ndi matenda mu ndondomeko magazi. Komanso, mankhwala kuli ndi ubwino pa thupi la munthu ndi kupweteka kwa mutu, senile maganizo ndi zinthu pambuyo sitiroko.
Tiyenera kuona kuti wothandizila ankaona zimayambitsa zochita mbali. Pofuna kupewa chitukuko, ayenera kutsatira malangizo onse a dokotala. Tengani mapiritsi "tsinarin" nzeru zake yekha, adzathetsedwa. Iwo ayenera mankhwala okha ndi dokotala nawo.
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