Thanzi, Kukonzekera
Drotaverina hydrochloride
hydrochloride Drotaverina chikukhudza nyimbo mankhwala ndi zotsatira spasmolytic. ntchito zake walangizidwa minofu yosalala ya m'mimba ziwalo, urogenital ndi biliary dongosolo, komanso mtima yosalala minofu wosanjikiza. Drotaverina hydrochloride (Nospanum), kulimbikitsa zosangalatsa zigawo yosalala minofu, ndi okhoza kuthetsa cramping. Komanso, mankhwala bwino minofu zakudya mpweya ndi yowonjezera mtima lumen. Drotaverina hydrochloride amatha kusintha angathe selo nembanemba ndi permeability. The medicament amachepetsa ntchito enzymatic wa phosphodiesterase, kukwezeletsa zikugwilizana (yunifolomu) kuonjezera msasa misinkhu ndi mayamwidwe koyamba kwa maselo kashiamu ion.
Drotaverina hydrochloride yodziwika ndi digiri otsika lumikiza ndi mapuloteni plasma. Kwambiri ndichifukwa chimamanga kuti beta ndi alpha-globulins, albumin. Pasanathe mphindi makumi asanu ndi makumi asanu ndi limodzi pambuyo makonzedwe m'kamwa madzi a m'magazi ntchito kuwawonetsera ndende nsonga ya thunthu yogwira. Hafu ya moyo wa dongosolo la maola makumi awiri ndi ziwiri. Excretion wa metabolites amapangidwa makamaka mu mkodzo. Part wa excretion wa mankhwala akupezeka ndowe za.
The medicament (mu mawonekedwe a njira jekeseni, ndi miyala) akapatsidwa kuthetsa mpumulo ululu chonsechi chikhalidwe ndi kuphipha. hydrochloride Drotaverina zikusonyeza chapamimba chilonda, cholecystitis, kudzimbidwa, chonsechi etiology, pyloric yosalala minofu kuphipha ndipo kadinala chapamimba khadi, cystitis, nephrolithiasis, proctitis, pyelitis ndi uretrolitiaze. Mankhwala ntchito omangana m'mimba chifukwa cha mpweya mwamsanga ndi chonsechi matenda a m'matumbo. medicament The Angagwiritsidwenso ntchito pochititsa diagnostics, kuphatikizapo holetsistografii lapansi. Drotaverine tapatsidwa vasodilatation ku chizindikiritso cha mtima minofu yosalala spasms wosanjikiza remover mutu kuphipha ziwiya ubongo. mankhwala kawirikawiri amagwiritsidwa ntchito algodismenoree kuchita matenda. The medicament ndi kuteteza ndi kuthetsa minofu yosalala omangana mu chiberekero pa mimba ndi nkhani ya kuopseza mimba. Iwo anasonyezanso mu nthawi yobereka kwa spasmolysis ndi protracted Kuwulura uterine pakhosi ndi pa ayi postnatal.
Drotaverina hydrochloride. Malangizo.
kukonzekera A mu mawonekedwe a mapiritsi kumwedwa pakamwa. Mapiritsi sayenera fodya ameneyu amatafunidwa kapena kum'pondereza, ayenera chimezedwe lonse, ndi madzi zedi okwanira. Mankhwala sikudalira pa nthawi ya chakudya. Mlingo ndi nthawi ya mankhwala anatsimikiza aliyense payekha ndi dokotala nawo.
Achinyamata (pa khumi ndi ziwiri) ndi akulu kuthetsa ululu chonsechi anaika mapiritsi 1-2 (40-80 mg) kawiri kapena katatu pa tsiku.
Ana osaposera zaka khumi kukonzekera wapatsidwa malinga ndi atasankhidwa dokotala.
The medicament mu mawonekedwe a jekeseni wa chikuyendetsedwera intramuscularly. Kwa odwala ndi insufficiency aimpso kapena kwa chiwindi, mwina m'mbuyo kumayambiriro mankhwala kudzera m'mitsempha. Njira imeneyi imagwira chomveka pokhapokha kukhazikitsidwa kwa malo yopingasa wodwala. Mu zotumphukira magazi chisokonezo chimene chayambitsa ndi mtima yosalala minofu kuphipha wosanjikiza kukhala wodekha intraarterial utsogoleli.
Monga ulamuliro, odwala kulekerera mankhwala. Komabe, nthawi zina, pangakhale mavuto. Mwachitsanzo, odwala akhoza kukhala nseru, mkhutu chopondapo, kusanza. Kumachitika, ndipo CNS matenda, monga kuphwanya maso ndi mode mpumulo (kugona), kupweteka kwa mutu, kukomoka. Panali milandu matenda a dongosolo mtima, anaonetsa tachycardia, arrhythmias, kutsitsa zoipazi. N'zothekanso kutupa kwa amphuno mucosa, thupi lawo siligwirizana, bronchospasm.
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